Mu opioid receptor antagonist 3

MedChem Express

Mu opioid receptor antagonist 3

10

Research Use Only

C25H28N2O4S

452.57

Mu opioid receptor antagonist 3 (compound 26) is a potent and selective micro opioid receptor (MOR) antagonist with a K i of 0.24 nM and an EC 50 of 0.54 nM. Mu opioid receptor antagonist 3 has remarkable CNS antagonism against morphine, and precipitated fewer withdrawal symptoms than Naloxone. Mu opioid receptor antagonist 3 can be used for researching opioid use disorders (OUD) [1] .

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