Omarigliptin (MK-3102) [1226781-44-7]
S8565
CAS Number1226781-44-7
Product group Chemicals
Overview
- SupplierSelleck Chemicals
- Product NameOmarigliptin (MK-3102) [1226781-44-7]
- Delivery Days Customer9
- CAS Number1226781-44-7
- CertificationResearch Use Only
- Scientific DescriptionOmarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 muM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 muM at IKr, Cagamma1.2, and Nagamma1.5).
- UNSPSC12352200