Pelabresib

MedChem Express

Pelabresib

14

Research Use Only

99.95

C20H16ClN3O2

365.81

Pelabresib (CPI-0610) is a potent, selective, orally active and cell-active BET inhibitor. Pelabresib inhibits BRD4-BD1 with an IC 50 of 39 nM, and with an EC 50 value of 0.18 microM for MYC [1] .

O=C(N)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C3=CC=CC=C3C4=C1ON=C4C

-20°C,2°C to 8°C

12352200