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PPARalpha/gamma agonist 5

Research Use Only
HY-167950
MedChem Express
Molecular Weight437.51
Product group Chemicals
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Overview

  • Supplier
    MedChem Express
  • Product Name
    PPARalpha/gamma agonist 5
  • Delivery Days Customer
    9
  • Certification
    Research Use Only
  • Molecular Formula
    C24H23NO5S
  • Molecular Weight
    437.51
  • Scientific Description
    PPARalpha/gamma agonist 5 is a dual PPARalpha/gamma agonist with significant biological activity exhibited at low concentrations. The EC50 of PPARalpha/gamma agonist 5 are 0.358microM and 1.21microM respectively, showing its potential in inhibiting type 2 diabetes and lipid metabolism disorders. PPARalpha/gamma agonist 5 was selected for clinical development due to its high efficacy[1].
  • SMILES
    OC([C@H](OC)CC1=C2C(C=CS2)=C(C=C1)OCCC3=C(C)OC(C4=CC=CC=C4)=N3)=O
  • UNSPSC
    12352200