PQ-69

MedChem Express

PQ-69 [910045-32-8]

10

910045-32-8

Research Use Only

C20H19FN4O

350.39

PQ-69 is a potent and selective adenosine A1 receptor antagonist with inverse agonist activity. PQ-69 binds to hA1 receptor with a K i value of 0.96 nM, is 217-fold more selective compared with hA2A receptors (K i =208 nM) and >1,000-fold selectivity over hA3 receptor (K i >100 microM). PQ-69 can be used for the research of renal dysfunction [1] .

O=C1N(C2=CC=CC(F)=C2)NC3=C1C(NCCCC)=NC4=CC=CC=C34

12352200