Protease-Activated Receptor-1 antagonist 3

MedChem Express

Protease-Activated Receptor-1 antagonist 3

10

Research Use Only

C30H34N4O3

498.62

Protease-Activated Receptor-1 antagonist 3 is a potent protease-activated receptor-1 antagonist with an IC50 value of 7 nM. Protease-Activated Receptor-1 antagonist 3 shows binding affinity for hERG K+ channel with an IC50 value of 9 microM[1].

[H][C@]12[C@H]([C@@H]([C@@H](C)[C@H]3[C@]1(C(O[C@@H]2C)=O)CN(C(NCC)=O)C3)C)/C=C/C4=CC=C(C=N4)C5=CC=CC=C5C#N

12352200