(Rac)-Telinavir
HY-106395A
Molecular Weight604.74
Product group Chemicals
Overview
- SupplierMedChem Express
- Product Name(Rac)-Telinavir
- Delivery Days Customer9
- CertificationResearch Use Only
- Molecular FormulaC33H44N6O5
- Molecular Weight604.74
- Scientific Description(Rac)-Telinavir ((Rac)-SC-52151) is a potent, selective, tight-binding human immunodeficiency virus (HIV) protease inhibitor that exhibits significant anti-HIV activity. (Rac)-Telinavir has a mean 50% effective concentration of 26 ng/ml (43 nM) against various strains of HIV, including HIV-1, HIV-2, and simian immunodeficiency virus. (Rac)-Telinavir, in combination with nucleoside reverse transcriptase inhibitors, demonstrates synergistic effects on inhibiting HIV-1 replication without additive toxicity. (Rac)-Telinavir is highly protein bound in human plasma and exhibits low partitioning into erythrocytes.
- SMILESO=C(CC(C(NC(C(CN(CC(C)C)C(NC(C)(C)C)=O)O)CC1=CC=CC=C1)=O)NC(C2=CC=C3C=CC=CC3=N2)=O)N
- UNSPSC12352200