rel-Delequamine

MedChem Express

rel-Delequamine

9

Research Use Only

C18H26N2O3S

350.48

rel-Delequamine (rel-RS-15385-197) is an orally active, brain-penetrant, potent and selective M 2 -adrenoceptor antagonist and alpha 2 -adrenoceptor antagonist. rel-Delequamine has a pK i of 9.45 for alpha 2 -adrenoceptors in the rat cortex. rel-Delequamine augments K + -evoked release of noradrenaline with an EC 50 of 1 nM [1] .

O=S(N1CCC[C@@]2(CN([C@]3(C[C@]12[H])[H])CCC4=C3C=CC(OC)=C4)[H])(C)=O

12352200