RK-701

MedChem Express

RK-701

10

Research Use Only

98.04

C26H30N4O3

446.54

RK-701 is an highly selective and non-genotoxic inhibitor of G9a with IC 50 value of 23-27 nM. RK-701 selectively up-regulates HbF, gamma- Globin, BGLT3 expression, down-regulates H3K9me2 expression. RK-701 also has inhibition for BCL11A and ZBTB7A [1] .

CC1=C(C(N[C@@H](CCC2CC2)C(NC3=CC=C(C=C3)C#N)=O)=O)NC(CC(C)(C4)C)=C1C4=O

-20°C,2°C to 8°C

12352200