RS 39604

MedChem Express

RS 39604 [167710-87-4]

10

167710-87-4

Research Use Only

98.0

C26H37Cl2N3O6S

590.56

RS 39604 is a potent, selective, and orally active 5-HT 4 receptor antagonist with a pK i of 9.1 in guinea pig striatal membranes. RS 39604 displays a low affinity (pK i 1A , 5-HT 2C , 5-HT 3 , alpha 1c , D 1 , D 2 , M 1 , M 2 , AT 1 , B 1 and opioid mu receptors and moderate affinity for delta 1 , (pK i =6.8) and delta 2 (pK i =7.8) sites [1] .

CS(=O)(NCCN1CCC(CCC(C2=CC(Cl)=C(N)C=C2OCC3=CC(OC)=CC(OC)=C3)=O)CC1)=O.Cl

2°C to 8°C

12352200