Ruboxistaurin [169939-94-0]

TargetMol Chemicals

Ruboxistaurin [169939-94-0]

114

169939-94-0

Chemical

Research Use Only

Ruboxistaurin

C28H28N4O3

468.55

Ruboxistaurin (LY333531) is a selective, orally active PKC beta inhibitor with a Ki value of 2 nM. Ruboxistaurin competitively inhibits PKC beta I (IC50: 4.7 nM) in an ATP-dependent manner. Ruboxistaurin is able to act on PKC beta II (IC50: 5.9 nM).

3 years

CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21

-20°C

12352200