TCS 1102 [916141-36-1]

MedChem Express

TCS 1102 [916141-36-1]

10

916141-36-1

Research Use Only

99.73

C27H26N4O2S

470.59

TCS 1102 is a potent, dual orexin receptor antagonist, with Ki values of 0.2 nM and 3 nM for OX2 and OX1 receptors, respectively. TCS 1102 demonstrates excellent blood-brain barrier penetrability and moderate bioavailability in rats[1].

O=C([C@H]1N(C(CSC2=NC3=CC=CC=C3N2C)=O)CCC1)NC4=CC=CC=C4C5=CC=CC=C5

-20°C,2°C to 8°C

12352200