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TG4-155 [1164462-05-8]

Research Use Only
HY-18971
MedChem Express
CAS Number1164462-05-8
Product group Chemicals
Estimated Purity99.91
Molecular Weight394.46
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Overview

  • Supplier
    MedChem Express
  • Product Name
    TG4-155 [1164462-05-8]
  • Delivery Days Customer
    10
  • CAS Number
    1164462-05-8
  • Certification
    Research Use Only
  • Estimated Purity
    99.91
  • Molecular Formula
    C23H26N2O4
  • Molecular Weight
    394.46
  • Scientific Description
    TG4-155 is a potent, brain-permeant and selective EP2 receptor antagonist with a Ki of 9.9 nM[1][2]. TG4-155 shows low nanomolar antagonist activity against only EP2 and DP1[1]. TG4-155 has an EP2 Schild KB of 2.4 nM and displays 550-4750-fold selectivity for EP2 over EP1, EP3, EP4 and IP, but only 14-fold selectivity against the DP1 receptor[2].
  • SMILES
    O=C(NCCN1C(C)=CC2=C1C=CC=C2)/C=C/C3=CC(OC)=C(OC)C(OC)=C3
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200