Torkinib (PP242)
ORB181304
CAS Number1092351-67-1
Product group Chemicals
Molecular Weight308.34
Overview
- SupplierBiorbyt
- Product NameTorkinib (PP242) [1092351-67-1]
- Delivery Days Customer16
- CAS Number1092351-67-1
- CertificationResearch Use Only
- Molecular FormulaC16H16N6O
- Molecular Weight308.34
- Scientific DescriptionPP242 is a selective mTOR inhibitor with IC50 of 8 nM; targets both mTOR complexes with > 10- and 100-fold selectivity for mTOR than PI3Kdelta or PI3Kalpha/beta/gamma, respectively; also showed slightly weaker activity against BRD4 (Kd= 1.7 uM).
- SMILESN1C2=C(C=C(O)C=C2)C=C1C1C2=C(N)N=CN=C2N(C(C)C)N=1
- UNSPSC12352200