TPOP146

Biorbyt

TPOP146 [2018300-62-2]

16

2018300-62-2

Research Use Only

C27H35N3O5

481.58

TPOP146 is a selective CBP/P300 benzoxazepine bromodomain inhibitor with Kd values of 134 nM and 5.02 microM for CBP and BRD4.

COC1=CC(OC)=CC(C2=CC(C(N[C@H]3CCCN(C)C3)=O)=C(OCCN(C(CC)=O)C4)C4=C2)=C1

12352200