Uzansertib

MedChem Express

Uzansertib [1620012-39-6]

10

1620012-39-6

Research Use Only

C26H26F3N5O3

513.51

Uzansertib (INCB053914) is an orally active, ATP-competitive pan- PIM kinase inhibitor with IC 50 s of 0.24 nM, 30 nM, 0.12 nM for PIM1, PIM2, PIM3, respectively. Uzansertib has broad anti-proliferative activity against a variety of hematologic tumor cell lines [1] .

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