Vicriviroc (malate)

MedChem Express

Vicriviroc (malate) [541503-81-5]

9

541503-81-5

Research Use Only

C32H44F3N5O7

667.72

Vicriviroc (SCH 417690) malate is an orally active CCR5 antagonist with the IC 50 of 10 nM, and also inhibts MIP-1alpha and intracellular calcium release induced by the ligand RANTES (10 nM) with the IC 50 values of 0.91 nM and 16 nM, respectively. Vicriviroc malate can inhibits human immunodeficiency virus type 1 (HIV-1) infection, and can also used for study of cancer [1] [2] .

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