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VUF10166

HY-100552
MedChem Express
CAS Number155584-74-0
Product group Chemicals
Estimated Purity99.83
Molecular Weight262.744
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Overview

  • Supplier
    MedChem Express
  • Product Name
    VUF10166 [155584-74-0]
  • Delivery Days Customer
    10
  • CAS Number
    155584-74-0
  • Estimated Purity
    99.83
  • Molecular Formula
    C13H15ClN4
  • Molecular Weight
    262.744
  • Scientific Description
    VUF10166 is a potent and high-affinity 5-HT 3 receptor antagonist, with K i values of 0.04 nM (5-HT 3 A) and 22 nM (5-HT 3 AB). VUF10166 inhibits 5-HT-induced responses at 5-HT 3 A and 5-HT 3 AB receptors at nanomolar concentrations. At 5-HT 3 receptor , VUF10166 at higher concentrations also acts as a partial agonist, with an EC 50 of 5.2 microM [1] .
  • SMILES
    CN1CCN(C2=NC3=CC=CC=C3N=C2Cl)CC1
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200