VUF10166
HY-100552
CAS Number155584-74-0
Product group Chemicals
Estimated Purity99.83
Molecular Weight262.744
Overview
- SupplierMedChem Express
- Product NameVUF10166 [155584-74-0]
- Delivery Days Customer10
- CAS Number155584-74-0
- Estimated Purity99.83
- Molecular FormulaC13H15ClN4
- Molecular Weight262.744
- Scientific DescriptionVUF10166 is a potent and high-affinity 5-HT 3 receptor antagonist, with K i values of 0.04 nM (5-HT 3 A) and 22 nM (5-HT 3 AB). VUF10166 inhibits 5-HT-induced responses at 5-HT 3 A and 5-HT 3 AB receptors at nanomolar concentrations. At 5-HT 3 receptor , VUF10166 at higher concentrations also acts as a partial agonist, with an EC 50 of 5.2 microM [1] .
- SMILESCN1CCN(C2=NC3=CC=CC=C3N=C2Cl)CC1
- Storage Instruction2°C to 8°C
- UNSPSC12352200