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YM-230888

HY-107510
MedChem Express
CAS Number446257-23-4
Product group Chemicals
Molecular Weight360.52
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Overview

  • Supplier
    MedChem Express
  • Product Name
    YM-230888
  • Delivery Days Customer
    9
  • CAS Number
    446257-23-4
  • Certification
    Research Use Only
  • Molecular Formula
    C19H28N4OS
  • Molecular Weight
    360.52
  • Scientific Description
    YM-230888 is an orally active, selective and allosteric mGlu1 receptor antagonist with a K i of 13 nM. YM-230888 inhibits mGlu1-mediated inositol phosphate production in rat cerebellar granule cells with an IC 50 of 13 nM. YM-230888 shows antinociceptive response in Streptozotocin (HY-13753)-induced hyperalgesia models. YM-230888 significantly reduces pain parameters in complete Freunds adjuvant (HY-153808)-induced arthritic pain models [1] .
  • SMILES
    C1(NC2CCCCCC2)=C3C(SC(CNC[C@H]4CCCO4)=C3)=NC=N1
  • UNSPSC
    12352200