Zanoterone

MedChem Express

Zanoterone

5

Research Use Only

C23H32N2O3S

416.58

Zanoterone is an orally active antagonist of the androgen receptor (AR) with a K i of 2.2 microM. Zanoterone blocks the binding of androgens such as testosterone and dihydrotestosterone (DHT), inhibiting the androgen signaling pathway, thereby reducing androgen-dependent prostate hyperplasia and prostate cancer growth [1] .

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