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2-Amino-6-chloropurine-9-(2-O-propargyl)riboside [2095417-35-7]

HY-152746
MedChem Express
Product group Molecular Biology
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Overview

  • Supplier
    MedChem Express
  • Product Name
    2-Amino-6-chloropurine-9-(2-O-propargyl)riboside [2095417-35-7]
  • Delivery Days Customer
    10
  • CAS Number
    2095417-35-7
  • Certification
    Research Use Only
  • Molecular Formula
    C13H14ClN5O4
  • Molecular Weight
    339.73
  • Scientific Description
    2-Amino-6-chloropurine-9-(2-O-propargyl)riboside is a purine nucleoside analogue. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc[1]. 2-Amino-6-chloropurine-9-(2-O-propargyl)riboside is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
  • SMILES
    O[C@H]1[C@@H](OCC#C)[C@H](N(C=N2)C3=C2C(Cl)=NC(N)=N3)O[C@@H]1CO
  • UNSPSC
    41115811