3-Bromocytisine

MedChem Express

3-Bromocytisine [207390-14-5]

10

207390-14-5

Research Use Only

99.90

C11H13BrN2O

269.14

3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, with IC 50 s are 0.28, 0.30 and 31.6 nM for halpha4beta4, halpha4beta2, and halpha7-nACh, respectively. 3-Bromocytisine (3-Br-cytisine) shows different effects on high (HS) and low (LS) ACh sensitivity alpha4beta2 nAChRs with EC 50 s are 8 and 50 nM, respectively [1] [2] .

O=C1N2C([C@]3([H])C[C@](CNC3)([H])C2)=CC=C1Br

-20°C

12352200