3-Hydroxy darifenacin [206048-82-0]

MedChem Express

3-Hydroxy darifenacin [206048-82-0]

5

206048-82-0

Research Use Only

C28H30N2O3

442.55

3-Hydroxy darifenacin is a metabolite of Darifenacin (HY-A0033). 3-Hydroxy darifenacin is an antagonist of M1-5 muscarinic receptors with Kis values of 17.78, 79.43, 2.24, 36.31 and 6.17 nM, respectively in CHO cells[1].

NC(C(C1=CC=CC=C1)(C2=CC=CC=C2)[C@H]3CN(CC3)CCC4=CC=C(OCC5O)C5=C4)=O

12131703