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4-Epianhydrochlortetracycline (hydrochloride) [158018-53-2]

HY-120715
MedChem Express
CAS Number158018-53-2
Product group Chemicals
Molecular Weight497.33
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Overview

  • Supplier
    MedChem Express
  • Product Name
    4-Epianhydrochlortetracycline (hydrochloride) [158018-53-2]
  • Delivery Days Customer
    5
  • CAS Number
    158018-53-2
  • Certification
    Research Use Only
  • Molecular Formula
    C22H22Cl2N2O7
  • Molecular Weight
    497.33
  • Scientific Description
    4-Epianhydrochlortetracycline hydrochloride is an inhibitor of matrix metalloproteinases (MMPs), particularly gelatinase B (Gelatinase B, EC 3.4.24.35), with inhibition rates of 100% at 500 microg/mL, 70% at 125 microg/mL, and 40% at 31 microg/mL. 4-Epianhydrochlortetracycline hydrochloride is promising for research in chronic inflammatory diseases[1].
  • SMILES
    O[C@]12[C@](CC(C(C2=O)=C(C3=C(O)C=C4)O)=C(C)C3=C4Cl)([H])[C@H](C(O)=C(C1=O)C(N)=O)N(C)C.Cl
  • UNSPSC
    12352200