A1/A3 AR antagonist 1

MedChem Express

A1/A3 AR antagonist 1 [312929-49-0]

10

Research Use Only

C24H18N2O3S

414.48

A1/A3 AR antagonist 1 (compound 10) is a potent adenosine 1 (A1) and adenosine 3 (A3) receptor dual antagonist with Kis of 36.7 nM, 25.4 nM and 1.47 nM for human A1, human A3 and rat A1, respectively. A1/A3 AR antagonist 1 can be used for researching kidney failure, inflammatory pulmonary diseases, and Alzheimers disease[1].

COC1=CC=C(C=C1)C(NC2=NC(C3=CC=CC=C3)=C(S2)C(C4=CC=CC=C4)=O)=O

12131703