A2A receptor antagonist 3 [2738606-83-0]

MedChem Express

A2A receptor antagonist 3 [2738606-83-0]

5

2738606-83-0

Research Use Only

C26H26N6O2

454.52

A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist with a Ki of 0.4 nM. A2A receptor antagonist 3 also binds to A2b, A1 and A3 receptor with Kis of 37, 107 and 1467 nM, respectively[1].

CC(C)(O)[C@H](C)NC(C1=NC2=C(C3=CC(C)=NC(C)=C3)C(C4=CC(C#N)=CC=C4)=NN2C=C1)=O

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