A2A/A3 AR antagonist-1

MedChem Express

A2A/A3 AR antagonist-1 [1448221-36-0]

10

Research Use Only

C56H71N15O12S2

1210.39

A2A/A3 AR antagonist-1 (compound 23) is a dual A2A/A3 adenosine receptor (AR) fluorescent ligand, with Kis of 90 nM and 31.8 nM for hA2A AR and hA3 AR, respectively[1].

CN1C=C2C(N=C(N3N=C(N=C23)C4=CC=CO4)NC(CCCC5=CN(N=N5)CCCCCCNC(C6=CC(C([O-])=O)=C(C=C6)C7=C8C=CC(C(S(=O)([O-])=O)=C8OC9=C(C(N)=CC=C97)S(=O)([O-])=O)=[NH2+])=O)=O)=N1.CC[NH+](CC)CC.CC[NH+](CC)CC

12131703