A3AR antagonist 3 [863202-33-9]

MedChem Express

A3AR antagonist 3 [863202-33-9]

14

863202-33-9

Research Use Only

C17H18N6

306.37

A3AR antagonist 3 (compound 21) is a selective A3 adenosine receptor (A3AR) antagonist with a Ki of 37 nM. A3AR antagonist 3 shows >60-fold selectivity in comparison to A1 and A2A adenosine receptors[1].

[H][C@@]12[C@H]([C@@](C2)([H])CC1)NC3=C4N=CNC4=NC(NC5=CC=CC=C5)=N3

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