AG-041R

MedChem Express

AG-041R [159883-95-1]

5

159883-95-1

Research Use Only

C31H36N4O5

544.64

AG-041R is a potent and selective CCK2 Receptor/Gastrin antagonist. AG-041R inhibits gastrin-evoked secretion of pancreastatin with an IC 50 of 2.2 nM. AG-041R inhibits cell growth of Mastomys ECL carcinoid tumor cells [1] [2] .

CC(C=C1)=CC=C1NC(C[C@]2(C3=CC=CC=C3N(C2=O)CC(OCC)OCC)NC(NC4=CC=C(C=C4)C)=O)=O

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