Bio-Connect

AKR1C2/3-IN-2 [56600-73-8]

HY-121656
MedChem Express
CAS Number56600-73-8
Product group Chemicals
Molecular Weight244.29
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Overview

  • Supplier
    MedChem Express
  • Product Name
    AKR1C2/3-IN-2 [56600-73-8]
  • Delivery Days Customer
    9
  • CAS Number
    56600-73-8
  • Certification
    Research Use Only
  • Molecular Formula
    C15H16O3
  • Molecular Weight
    244.29
  • Scientific Description
    AKR1C2/3-IN-2 is a potential AKR1C3 inhibitor with selective AKR1C3 activity. AKR1C2/3-IN-2 is able to block AKR1C3-mediated testosterone (T) production and PSA induction, affecting the endocrine activity of prostate cancer cells. AKR1C2/3-IN-2 shows selectivity over other AKR1C enzymes, indicating its potential application in inhibiting drug-resistant prostate cancer. AKR1C2/3-IN-2 has no inhibitory activity against COX isomerases, further emphasizing its specificity as a prostate cancer inhibitory compound[1].
  • SMILES
    O=C(C(CC)C1=CC=C2C=C(C=CC2=C1)OC)O
  • UNSPSC
    12352200