AKR1C2/3-IN-2 [56600-73-8]
HY-121656
CAS Number56600-73-8
Product group Chemicals
Molecular Weight244.29
Overview
- SupplierMedChem Express
- Product NameAKR1C2/3-IN-2 [56600-73-8]
- Delivery Days Customer9
- CAS Number56600-73-8
- CertificationResearch Use Only
- Molecular FormulaC15H16O3
- Molecular Weight244.29
- Scientific DescriptionAKR1C2/3-IN-2 is a potential AKR1C3 inhibitor with selective AKR1C3 activity. AKR1C2/3-IN-2 is able to block AKR1C3-mediated testosterone (T) production and PSA induction, affecting the endocrine activity of prostate cancer cells. AKR1C2/3-IN-2 shows selectivity over other AKR1C enzymes, indicating its potential application in inhibiting drug-resistant prostate cancer. AKR1C2/3-IN-2 has no inhibitory activity against COX isomerases, further emphasizing its specificity as a prostate cancer inhibitory compound[1].
- SMILESO=C(C(CC)C1=CC=C2C=C(C=CC2=C1)OC)O
- UNSPSC12352200