Bio-Connect

AKT-IN-VIII [612847-09-3] [612847-09-3]

BS-6708C
Bioss
CAS Number612847-09-3
Product group Chemicals
Estimated Purity98 - 98.0
Molecular Weight551.64
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Overview

  • Supplier
    Bioss
  • Product Name
    AKT-IN-VIII [612847-09-3] [612847-09-3]
  • Delivery Days Customer
    16
  • CAS Number
    612847-09-3
  • Certification
    Research Use Only
  • Conjugate
    Unconjugated
  • Estimated Purity
    98 - 98.0
  • Molecular Formula
    C34 H29 N7 O
  • Molecular Weight
    551.64
  • Scientific Description
    AKT-IN-VIII, also known as AKTi-1/2, is a potent, selective and ell permeable, allosteric inhibitor of Akt 1 and 2, which efficiently inhibits CaMKIalpha activity and aryl hydrocarbon receptor pathway. AKT-IN-VIII suppresses hyperthermia-induced Ndrg2 phosphorylation in gastric cancer cells. AKT-IN-VIII displays good selectivity against a panel of 70 other kinases with micromolar inhibition against some kinases, for example, calcium/calmodulin-dependent protein kinase 1 and smooth muscle myosin light-chain kinase.
  • SMILES
    O=C1NC2C=CC=CC=2N1C1CCN(CC2C=CC(=CC=2)C2N=C3C=C4NC=NC4=CC3=NC=2C2C=CC=CC=2)CC1
  • Storage Instruction
    -20°C
  • UNSPSC
    12161509