Apabetalone

MedChem Express

Apabetalone [1044870-39-4]

10

1044870-39-4

Research Use Only

99.47

C20H22N2O5

370.40

Apabetalone (RVX-208) is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. The IC 50 s are 87 microM and 0.51 microM for BD1 and BD2 , respectively [1] .

COC1=CC(OC)=C(C(NC(C2=CC(C)=C(OCCO)C(C)=C2)=N3)=O)C3=C1

-20°C,2°C to 8°C

12352200