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ARC 239 (dihydrochloride) [55974-42-0]

HY-12709A
MedChem Express
CAS Number55974-42-0
Product group Chemicals
Estimated Purity99.20
Molecular Weight480.43
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Overview

  • Supplier
    MedChem Express
  • Product Name
    ARC 239 (dihydrochloride) [55974-42-0]
  • Delivery Days Customer
    10
  • CAS Number
    55974-42-0
  • Certification
    Research Use Only
  • Estimated Purity
    99.20
  • Hazard Information
    h302, h400, h410
  • Molecular Formula
    C24H31Cl2N3O3
  • Molecular Weight
    480.43
  • Scientific Description
    ARC 239 dihydrochloride is a selective alpha2B/2C adrenoceptor antagonist (pKd values are 5.95, 7.41 and 7.56 at alpha2A, alpha2B, and alpha2C receptors respectively). ARC 239 dihydrochloride binds to CHO cell membranes expressing human recombinant a2A-, a2B- or a2C-adrenoceptor subtypes with pKis of 5.6, 8.4, and 7.08, respectively[1].
  • SMILES
    O=C1C2=C(C(C)(C)C(N1CCN3CCN(CC3)C4=C(OC)C=CC=C4)=O)C=CC=C2.Cl.Cl
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200