ARP-100 (Standard) [704888-90-4]

MedChem Express

ARP-100 (Standard) [704888-90-4]

5

Research Use Only

ARP-100 (Standard) is the analytical standard of ARP-100. This product is intended for research and analytical applications. ARP-100 is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM). ARP-100 interacts with S1 pocket of MMP-2 and shows anti-invasive properties in an in vitro model of invasion on matrigel. ARP-100 shows the less inhibitory activity towards MMP-1 (>50 microM), MMP-3 (4.5 microM), MMP-7 (>50 microM), and MMP-9 (0.2 microM)[1][2].

41116100