AST-1306 (TsOH)

AbMole BioScience

AST-1306 (TsOH)

9

1050500-29-2

Research Use Only

>99.0%

C24H18ClFN4O2

621.08

AST-1306 is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of 0.5 nM and 3 nM, also effective in mutation EGFR T790M/L858R, more potent to ErbB2-overexpressing cells, 3000-fold selective for ErbB family than other kinases,

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