Azepexole (dihydrochloride)

MedChem Express

Azepexole (dihydrochloride)

10

36067-72-8

Research Use Only

C9H17Cl2N3O

254.16

Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for alpha2A-, alpha2B- and alpha2C-adrenoceptor subtypes, resepctively[1]. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM)[2].

NC(O1)=NC2=C1CCN(CC)CC2.[H]Cl.[H]Cl

12352200