Bio-Connect

B026 [2379416-48-3]

HY-147261
MedChem Express
CAS Number2379416-48-3
Product group Chemicals
Molecular Weight557.50
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Overview

  • Supplier
    MedChem Express
  • Product Name
    B026 [2379416-48-3]
  • Delivery Days Customer
    10
  • CAS Number
    2379416-48-3
  • Certification
    Research Use Only
  • Molecular Formula
    C27H23F4N5O4
  • Molecular Weight
    557.50
  • Scientific Description
    B026 is a selective, potent, orally active p300/CBP histone acetyltransferase (HAT) inhibitor with IC50 values of 1.8 nM and 9.5 nM for p300 and CBP enzyme, respectively. B026 has anticancer activity for androgen receptor-positive (AR+) prostate cancer cell lines[1].
  • SMILES
    O=C1[C@@]2(NC(N1CC(N3[C@@H](COC4=CC=C(F)C=C4C3)C(F)(F)F)=O)=O)C5=CC=C(C6=CN(N=C6)C)C=C5CC2
  • UNSPSC
    12131703