BD-9136
HY-149878
Overview
- SupplierMedChem Express
- Product NameBD-9136 [3037514-38-5]
- Delivery Days Customer14
- CertificationResearch Use Only
- Estimated Purity98.81
- Molecular FormulaC44H44N10O5S
- Molecular Weight824.95
- Scientific DescriptionBD-9136 is a potent and highly selective BRD4 PROTAC depressant. BD-9136 has low-nanomolar degradation potencies against BRD4 , and its degradation selectivity for BRD4 is 1000 times that of BRD2 and BRD3 proteins. BD-9136 has antitumor activity[1].(Pink: Desmethyl-QCA276 (HY-44103); Black: 3-(2-(4-Methylpiperazin-1-yl)ethyl)azetidin-3-ol; Blue: Thalidomide-4-OH (HY-103596))
- SMILESCC1=NN=C2COCC(C(CC3=CC=CC=C3)=C(S4)C#CC5=CN(N=C5)C6(CCN7CCN(CC7)C)CN(C8=C(C9=CC=C8)C(N(C9=O)C%10CCC(NC%10=O)=O)=O)C6)=C4N21
- Storage Instruction-20°C
- UNSPSC12131703