BI-2081 [1458656-71-7]

MedChem Express

BI-2081 [1458656-71-7]

10

1458656-71-7

Research Use Only

C32H35FO6

534.62

BI-2081 is a GPR40 (FFAR1) partial agonist (EC50: 4 nM). BI-2081 induces glucose depending insulin secretion and reduces the plasma glucose concentration. BI-2081 can be used in the research of metabolic diseases, in particular diabetes type 2[1].

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