BI-3802

MedChem Express

BI-3802 [2166387-65-9]

10

2166387-65-9

Research Use Only

99.43

C24H29ClN6O3

484.98

BI-3802 is a highly potent BCL6 degrader and inhibits the Bric-a-brac (BTB) domain of BCL6 with an IC 50 of ≤3 nM. BI-3802 induces the polymerization of BCL6 and promotes BCL6 degration depended on E3 ligase SIAH1 . BI-3802 has antitumor activity [1] [2] .

ClC1=CN=C(N2C[C@H](C)C[C@H](C)C2)N=C1NC3=CC(C=C(OCC(NC)=O)C(N4C)=O)=C4C=C3

-20°C,2°C to 8°C

12352200