BI-D1870 [501437-28-1]

TargetMol Chemicals

BI-D1870 [501437-28-1]

4

501437-28-1

Chemical

Research Use Only

BI-D1870

99.43%

C19H23F2N5O2

391.42

BI-D1870 is a highly specific, blood-brain-permeable, and ATP-competitive inhibitor of the N-terminal AGC kinase domain of RSK, with IC50 values of 31 nM, 24 nM, 18 nM, and 15 nM for RSK1, RSK2, RSK3, and RSK4.

3 years

CC(C)CCN1C(C)C(=O)N(C)c2cnc(Nc3cc(F)c(O)c(F)c3)nc12

-20°C

12352200