BJJF078 [2531244-56-9]

MedChem Express

BJJF078 [2531244-56-9]

5

2531244-56-9

Research Use Only

99.34

C27H29N3O6S

523.60

BJJF078 is an aminopiperidine derivative. BJJF078 is a potent inhibitor of recombinant human and mouse Transglutaminase enzyme (TG2) activity, IC50 values of 41 and 54 nM, respectively. BJJF078 also inhibits the close related enzyme TG1, with an IC50 of 0.16 microM. BJJF078 can be used for Multiple sclerosis (MS) research[1].

O=C(NC1CCN(S(=O)(C2=C3C=CC=C(NC(C4=CC=C(C(OC)=C4)OC)=O)C3=CC=C2)=O)CC1)C=C

-20°C,2°C to 8°C

12131703