BMS-470539 (dihydrochloride) [2341796-82-3]
HY-115644
CAS Number2341796-82-3
Product group Chemicals
Estimated Purity99.85
Molecular Weight632.62
Overview
- SupplierMedChem Express
- Product NameBMS-470539 (dihydrochloride) [2341796-82-3]
- Delivery Days Customer10
- CAS Number2341796-82-3
- CertificationResearch Use Only
- Estimated Purity99.85
- Molecular FormulaC32H43Cl2N5O4
- Molecular Weight632.62
- Scientific DescriptionBMS-470539 dihydrochloride is a highly potent and selective melanocortin-1 receptor (MC-1R) agonist with an IC50 of 120 nM, an EC50 of 28 nM. BMS-470539 dihydrochloride does not activate MC-3R and is a very weak partial agonist at MC-4R and MC-5R. BMS-470539 dihydrochloride has potently anti-inflammatory properties[1][2][3].
- SMILESCCCC(C1(C2=CC=CC=C2)CCN(C([C@@H](CC3=CC=C(C=C3)OC)NC([C@H](CC4=CN=CN4C)N)=O)=O)CC1)=O.Cl.Cl
- Storage Instruction-20°C
- UNSPSC12352200
![BMS-470539 dihydrochloride [2341796-82-3]](https://www.targetmol.com/group3/M00/3F/0B/CgoaEWbYP6WEBN98AAAAAK3oiPs839.png)