Bio-Connect

BMS-470539 (dihydrochloride) [2341796-82-3]

HY-115644
MedChem Express
CAS Number2341796-82-3
Product group Chemicals
Estimated Purity99.85
Molecular Weight632.62
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Overview

  • Supplier
    MedChem Express
  • Product Name
    BMS-470539 (dihydrochloride) [2341796-82-3]
  • Delivery Days Customer
    10
  • CAS Number
    2341796-82-3
  • Certification
    Research Use Only
  • Estimated Purity
    99.85
  • Molecular Formula
    C32H43Cl2N5O4
  • Molecular Weight
    632.62
  • Scientific Description
    BMS-470539 dihydrochloride is a highly potent and selective melanocortin-1 receptor (MC-1R) agonist with an IC50 of 120 nM, an EC50 of 28 nM. BMS-470539 dihydrochloride does not activate MC-3R and is a very weak partial agonist at MC-4R and MC-5R. BMS-470539 dihydrochloride has potently anti-inflammatory properties[1][2][3].
  • SMILES
    CCCC(C1(C2=CC=CC=C2)CCN(C([C@@H](CC3=CC=C(C=C3)OC)NC([C@H](CC4=CN=CN4C)N)=O)=O)CC1)=O.Cl.Cl
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200