BMS-986187

MedChem Express

BMS-986187 [684238-37-7]

10

684238-37-7

Research Use Only

98.93

C31H34O4

470.60

BMS-986187 is an delta-opioid receptor -selective positive allosteric modulator (PAM) with an EC 50 of 0.03 microM and a pK B ?of 6.02 (~1?microM). BMS-986187 has no observable PAM activity at the?micro-receptor (EC 50 =3 microM) [1] .

CC1=C(C=CC=C1)COC2=CC=C(C=C2)C3C4=C(OC(CC(C)(C5)C)=C3C5=O)CC(C)(C)CC4=O

2°C to 8°C

12352200