BQ-788 (sodium salt)

MedChem Express

BQ-788 (sodium salt) [156161-89-6]

10

156161-89-6

99.33

C34H50N5NaO7

663.78

BQ-788 sodium salt is a potent and selective ETB receptor antagonist, inhibiting ET-1 binding to ETB receptors with an IC 50 of 1.2 nM in human Girrardi heart cells [1] .

CCCC[C@H](C(O[Na])=O)NC([C@@H](CC1=CN(C(OC)=O)C2=CC=CC=C12)NC([C@H](CC(C)(C)C)NC(N3[C@H](C)CCC[C@@H]3C)=O)=O)=O

-20°C

12352200