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BRK inhibitor P21d hydrochloride [2250025-98-8]

BRK inhibitor P21d hydrochloride [2250025-98-8]

T39772
TargetMol Chemicals
CAS Number2250025-98-8
Product group Chemicals
Molecular Weight483.93
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    BRK inhibitor P21d hydrochloride [2250025-98-8]
  • Delivery Days Customer
    86
  • CAS Number
    2250025-98-8
  • Certification
    Research Use Only
  • Chemical Name
    BRK inhibitor P21d hydrochloride
  • Molecular Formula
    C23H23ClFN7O2
  • Molecular Weight
    483.93
  • Scientific Description
    BRK inhibitor P21d hydrochloride is a highly potent inhibitor of breast tumor kinase (BRK/PTK6), displaying an IC50 of 30 nM, and effectively suppresses p-SAM68 with an IC50 of 52 nM. This compound serves as a valuable tool for evaluating BRK inhibitors efficacy in xenograft breast tumor models, enabling in vivo activity assessment.
  • Shelf life instruction
    3 years
  • SMILES
    Cl.Fc1cc(ccc1Nc1nc(cn2c(cnc12)-c1cn[nH]c1)C1CC1)C(=O)N1CCOCC1
  • Storage Instruction
    -20°C
  • UNSPSC
    51202000