Cavalpha2delta1&NET-IN-1 [2314361-39-0]
HY-148862
CAS Number2314361-39-0
Product group Chemicals
Molecular Weight422.54
Overview
- SupplierMedChem Express
- Product NameCavalpha2delta1&NET-IN-1 [2314361-39-0]
- Delivery Days Customer10
- CAS Number2314361-39-0
- CertificationResearch Use Only
- Molecular FormulaC23H26N4O2S
- Molecular Weight422.54
- Scientific DescriptionCavalpha2delta1&NET-IN-1 (Compound 59S) is a dual inhibitor of the alpha2delta-1 subunit of voltage-gated calcium channels (Cavalpha2delta-1) and the norepinephrine transporter (NET). Cavalpha2delta1&NET-IN-1 inhibits Cavalpha2delta-1 with a Ki of 112 nM. Cavalpha2delta1&NET-IN-1 inhibits NET with a Ki of 383 nM and IC50 of 67 nM. Cavalpha2delta1&NET-IN-1 can be used for research of pain[1].
- SMILESO=C1N(CCN(C2=NC=CC=C21)C)C3=CC(O[C@H](C4=CC=CS4)CCNC)=CC=C3
- UNSPSC12131703