Bio-Connect

Cavalpha2delta1&NET-IN-2 [2143586-17-6]

HY-148863
MedChem Express
CAS Number2143586-17-6
Product group Chemicals
Molecular Weight438.55
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Cavalpha2delta1&NET-IN-2 [2143586-17-6]
  • Delivery Days Customer
    10
  • CAS Number
    2143586-17-6
  • Certification
    Research Use Only
  • Molecular Formula
    C22H26N6O2S
  • Molecular Weight
    438.55
  • Scientific Description
    Cavalpha2delta1&NET-IN-2 (Compound 45CS) is a dual inhibitor of the alpha2delta-1 subunit of voltage-gated calcium channels (Cavalpha2delta-1) and the norepinephrine transporter (NET). Cavalpha2delta1&NET-IN-2 inhibits Cavalpha2delta-1 with a Ki of 454 nM. Cavalpha2delta1&NET-IN-2 inhibits NET with a Ki of 59 nM and IC50 of 7 nM. Cavalpha2delta1&NET-IN-2 can be used for research of pain[1].
  • SMILES
    O=C1N(CCN(C2=NC(N)=NC=C21)C)C3=CC(O[C@H](C4=CC=CS4)CCNC)=CC=C3
  • UNSPSC
    12131703