CAY10508
ORB2283712
CAS Number878533-35-8
Product group Chemicals
Estimated Purity98.00%
Molecular Weight486.2
Overview
- SupplierBiorbyt
- Product NameCAY10508
- Delivery Days Customer10
- CAS Number878533-35-8
- CertificationResearch Use Only
- Estimated Purity98.00%
- Molecular FormulaC21H14Br2N2O2
- Molecular Weight486.2
- Scientific DescriptionCAY10508 is a potent and selective inverse agonist for the central cannabinoid (CB1) receptor with therapeutic potential for treating obesity and drug dependence, lacking psychotropic effects. It exhibits a Ki value of 243 nM and an EC50 of 195 nM. At a concentration of 10 microM, CAY10508 displaces [3H]-CP-55,940 with 100% efficacy at the CB1 receptor and 35% at the peripheral cannabinoid (CB2) receptor. Its inverse agonist activity at the CB1 receptor was confirmed through a [35S]-GTPgammaS binding assay.
- SMILESO=C1C(N(C(=O)N1C2=CC=C(Br)C=C2)C3=CC=C(Br)C=C3)C4=CC=CC=C4
- Storage Instruction-20°C
- UNSPSC12352200
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