CB1/2 agonist 4 [2772949-38-7]
HY-150030
CAS Number2772949-38-7
Product group Chemicals
Molecular Weight431.65
Overview
- SupplierMedChem Express
- Product NameCB1/2 agonist 4 [2772949-38-7]
- Delivery Days Customer10
- CAS Number2772949-38-7
- CertificationResearch Use Only
- Molecular FormulaC27H45NO3
- Molecular Weight431.65
- Scientific DescriptionCB1/2 agonist 4 is a full CB1 agonist and CB2 partial agonist with EC50 values of 15.09 nM and 1.16 nM, respectively. CB1/2 agonist 4 also has hCB1 and hCB2 receptor affinities with Ki values of 1.1 nM and 4.2 nM, respectively. CB1/2 agonist 4 has a significant antinociceptive activity, and also can activate cannabinoid and TRPV1 receptor with values of IC50 and EC50 is 0.8 microM and 0.12 microM, respectively[1].
- SMILESO=C(NC1CC1)CCCCCCCOC2=CC(C(CCCCCC)(C)C)=CC(OC)=C2
- UNSPSC12131703