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CB1/2 agonist 4 [2772949-38-7]

HY-150030
MedChem Express
CAS Number2772949-38-7
Product group Chemicals
Molecular Weight431.65
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Overview

  • Supplier
    MedChem Express
  • Product Name
    CB1/2 agonist 4 [2772949-38-7]
  • Delivery Days Customer
    10
  • CAS Number
    2772949-38-7
  • Certification
    Research Use Only
  • Molecular Formula
    C27H45NO3
  • Molecular Weight
    431.65
  • Scientific Description
    CB1/2 agonist 4 is a full CB1 agonist and CB2 partial agonist with EC50 values of 15.09 nM and 1.16 nM, respectively. CB1/2 agonist 4 also has hCB1 and hCB2 receptor affinities with Ki values of 1.1 nM and 4.2 nM, respectively. CB1/2 agonist 4 has a significant antinociceptive activity, and also can activate cannabinoid and TRPV1 receptor with values of IC50 and EC50 is 0.8 microM and 0.12 microM, respectively[1].
  • SMILES
    O=C(NC1CC1)CCCCCCCOC2=CC(C(CCCCCC)(C)C)=CC(OC)=C2
  • UNSPSC
    12131703